Design, synthesis, antineoplastic activity of new pyrazolo[3,4-d]pyrimidine derivatives as dual CDK2/GSK3β kinase inhibitors; molecular docking study, and ADME prediction
Mohamed T. M. Nemr, Ahmed Elshewy, Mohammed L. Ibrahim, Ahmed M. El Kerdawy, Peter A. Halim
Topics & Concepts
ChemistryADMEPyrimidineDocking (animal)Combinatorial chemistryCyclin-dependent kinase 2StereochemistryKinaseBiochemistryProtein kinase AIn vitroNursingMedicineCancer-related Molecular PathwaysCancer Mechanisms and TherapyAdvanced Breast Cancer Therapies