Synthesis, antitumor, and apoptosis-inducing activities of novel 5-arylidenethiazolidine-2,4-dione derivatives: Histone deacetylases inhibitory activity and molecular docking study
Abdelrahman Hamdi, Walaa M. El-Husseiny, Dina I. A. Othman, Abdullah Haikal, Ahmed H. Bakheit, Adel S. El‐Azab, Mohamed H. Al‐Agamy, Alaa A.‐M. Abdel‐Aziz
Topics & Concepts
HDAC8ChemistryHDAC6Docking (animal)ApoptosisIC50CaspaseHDAC1Cell cycle checkpointHistoneCell culturePharmacologyCaspase 3Cell cycleBiochemistryStereochemistryHistone deacetylaseIn vitroProgrammed cell deathBiologyDNAGeneticsMedicineNursingHistone Deacetylase Inhibitors ResearchPeptidase Inhibition and AnalysisCholinesterase and Neurodegenerative Diseases