Discovery of small-molecule inhibitors of RUVBL1/2 ATPase
Gang Zhang, Feng Wang, Shan Li, Kai-Wen Cheng, Yingying Zhu, Ran Huo, Elyar Abdukirim, Guifeng Kang, Tsui‐Fen Chou
Topics & Concepts
ChemistryDocking (animal)PyrimidineSmall moleculeATPaseDrug discoveryStructure–activity relationshipEnzymeStereochemistryBiochemistryPharmacologyIn vitroBiologyNursingMedicineATP Synthase and ATPases ResearchBiochemical and Molecular ResearchUbiquitin and proteasome pathways