Balanced QSAR analysis to identify the structural requirements of ABBV-075 (Mivebresib) analogues as bromodomain and extraterminal domain (BET) family bromodomain inhibitor
Vijay H. Masand, Meghshyam K. Patil, Nahed N. E. El-Sayed, Magdi E. A. Zaki, Zainab M. Almarhoon, Sami A. Al‐Hussain
Topics & Concepts
ChemistryBromodomainQuantitative structure–activity relationshipStereochemistryCombinatorial chemistryComputational chemistryBiochemistryEpigeneticsGeneProtein Degradation and InhibitorsMultiple Myeloma Research and TreatmentsComputational Drug Discovery Methods