Design, synthesis and biological evaluation of potent EGFR kinase inhibitors against 19D/T790M/C797S mutation
Zhicheng Su, Tingyuan Yang, Jie Wang, Mengzhen Lai, Linjiang Tong, Gulinuer Wumaier, Zhuo Chen, Shengqing Li, Honglin Li, Hua Xie, Zhenjiang Zhao
Topics & Concepts
T790MChemistryKinasePharmacologyIC50EGFR inhibitorsCancer researchBiochemistryEpidermal growth factor receptorIn vitroReceptorBiologyGefitinibLung Cancer Treatments and MutationsCancer therapeutics and mechanismsHER2/EGFR in Cancer Research