Scaffold hopping of celastrol provides derivatives containing pepper ring, pyrazine and oxazole substructures as potent autophagy inducers against breast cancer cell line MCF-7
Feng Yao, Bing Zhang, Jialun Lv, Peng Zhang, Qing Mao, Fengwei Lin, Jiaxing Zhao, Xuefeng Fu, Yajun Yang, Zhaolin Li, Lei Zhang, Yanhua Mou, Shaojie Wang
Topics & Concepts
ChemistryMCF-7Cyclin-dependent kinaseCell cultureMTT assayAutophagyCancer cellCell growthCell cycle checkpointCell biologyCell cycleApoptosisCancer researchBiochemistryCancerHuman breastBiologyGeneticsNatural Compounds in Disease TreatmentAutophagy in Disease and TherapyCell death mechanisms and regulation