Design, synthesis and anticancer activities of novel dual poly(ADP-ribose) polymerase-1/histone deacetylase-1 inhibitors
Yongbin Tian, Zhouling Xie, Chenzhong Liao
Topics & Concepts
ChemistryPoly ADP ribose polymeraseOlaparibHistone deacetylasePARP inhibitorPharmacophorePolymeraseAcetylationPharmacologyStereochemistryBiochemistryHistoneEnzymeDNABiologyGenePARP inhibition in cancer therapyRadiation Effects in ElectronicsSemiconductor materials and devices