YC-1 potentiates the antitumor activity of gefitinib by inhibiting HIF-1α and promoting the endocytic trafficking and degradation of EGFR in gefitinib-resistant non-small-cell lung cancer cells
Hui Hu, Xiaokang Miao, Jingyi Li, Xiaowei Zhang, Jingjie Xu, Jingying Zhang, Tianxiong Zhou, Ming-Ning Hu, Wenle Yang, Lingyun Mou
Topics & Concepts
GefitinibCancer researchProtein kinase BEpidermal growth factor receptorTyrosine kinaseTyrosine-kinase inhibitorEGFR inhibitorsPharmacologyMedicineSignal transductionChemistryCancerInternal medicineBiochemistryGlycosylation and Glycoproteins ResearchLung Cancer Treatments and MutationsPeptidase Inhibition and Analysis