Litcius/Paper detail

Discovery of benzo[d]oxazol-2(3H)-one derivatives as a new class of TNIK inhibitors for the treatment of colorectal cancer

Xinling Luo, Ruicheng Yang, Yueshan Li, Liting Zhang, Shengyong Yang, Linli Li

2022Bioorganic & Medicinal Chemistry Letters10 citationsDOIOpen Access PDF

Topics & Concepts

Wnt signaling pathwayChemistryColorectal cancerIC50Drug discoveryCancer researchKinaseCancerWestern blotSignal transductionPharmacologyBiochemistryInternal medicineBiologyMedicineIn vitroGeneCancer-related Molecular PathwaysMechanisms of cancer metastasisCancer Mechanisms and Therapy