Synthesis of novel organohalogen chalcone derivatives and screening of their molecular docking study and some enzymes inhibition effects
Serdar Burmaoğlu, Elif Akın Kazancıoğlu, Rüya Kaya, Mustafa Zahrittin Kazancioğlu, Muhammet Karaman, Oztekin Algul, İlhami Gülçın
Topics & Concepts
ChalconeChemistryAcetylcholinesteraseCarbonic anhydraseEnzymeBiochemistryAchéDocking (animal)Active siteCarbonic Anhydrase IStereochemistryPharmacologyMedicineNursingEnzyme function and inhibitionPhenothiazines and Benzothiazines Synthesis and ActivitiesSynthesis and biological activity