Dual intra- and extracellular release of monomethyl auristatin E from a neutrophil elastase-sensitive antibody-drug conjugate
Imène Ait Mohamed Amar, Steve Huvelle, Emmanuel Douez, Stéphanie Letast, Sylvain Henrion, Marie‐Claude Viaud‐Massuard, Nicolas Aubrey, Émilie Allard-Vannier, Nicolas Joubert, Caroline Denevault‐Sabourin
Topics & Concepts
LinkerChemistryConjugateInternalizationAntibody-drug conjugateExtracellularIn vivoMonoclonal antibodyDrug deliveryIn vitroMechanism of actionPharmacologyBiochemistryAntibodyCellImmunologyBiologyOrganic chemistryComputer scienceMathematicsOperating systemBiotechnologyMathematical analysisHER2/EGFR in Cancer ResearchMonoclonal and Polyclonal Antibodies ResearchCell Adhesion Molecules Research