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Identification and Characterization of Two Structurally Related Dipeptides that Enhance Catalytic Efficiency of Neurolysin

Srinidhi Jayaraman, Joanna Kocot, Shiva Hadi Esfahani, Naomi J. Wangler, Arzu Uyar, Yehia Mechref, Paul C. Trippier, Thomas J. Abbruscato, Alex Dickson, Hideki Aihara, David A. Ostrov, Vardan T. Karamyan

2021Journal of Pharmacology and Experimental Therapeutics15 citationsDOIOpen Access PDF

Topics & Concepts

ChemistryPeptidomimeticDocking (animal)Combinatorial chemistryNeurotensinIn silicoSmall moleculeStereochemistryBiochemistryEnzymePeptideNeuropeptideReceptorGeneNursingMedicinePeptidase Inhibition and AnalysisNeuropeptides and Animal PhysiologyProtein Hydrolysis and Bioactive Peptides
Identification and Characterization of Two Structurally Related Dipeptides that Enhance Catalytic Efficiency of Neurolysin | Litcius