Evaluation of an ester-linked immunosuppressive payload: A case study in understanding the stability and cleavability of ester-containing ADC linkers
Courtney P. Jackson, Siteng Fang, Samantha R. Benjamin, Tchilabalo Dilezitoko Alayi, Yetrib Hathout, Sarah M. Gillen, Jillian P. Handel, Brittany M. Brems, Justin M. Howe, L. Nathan Tumey
Topics & Concepts
ChemistryCytosolInternalizationProdrugCatabolismBiochemistryCleaveCleavage (geology)LysosomeDeamidationEnzymeCellBiologyPaleontologyFracture (geology)Monoclonal and Polyclonal Antibodies ResearchHER2/EGFR in Cancer ResearchClick Chemistry and Applications