Quantitative estimation of drug permeation through nasal mucosa using in vitro membrane permeability across Calu-3 cell layers for predicting in vivo bioavailability after intranasal administration to rats
Daisuke Inoue, Tomoyuki Furubayashi, Akiko Tanaka, Toshiyasu Sakane, Kiyohiko Sugano
Topics & Concepts
BioavailabilityIn vivoNasal administrationPermeationPharmacologyMembrane permeabilityChemistryIn vitroPharmacokineticsDrugOral administrationMucous membrane of noseChromatographyMembraneMedicineImmunologyBiochemistryBiologyBiotechnologyAdvanced Drug Delivery SystemsDrug Transport and Resistance MechanismsDrug Solubulity and Delivery Systems