Litcius/Paper detail

Novel Peptidylarginine Deiminase Type 4 (PAD4) Inhibitors

Ram W. Sabnis

2022ACS Medicinal Chemistry Letters14 citationsDOIOpen Access PDF

Abstract

Provided herein are novel compounds as peptidylarginine deiminase type 4 (PAD4) inhibitors, pharmaceutical compositions, use of such compounds in treating diseases, and processes for preparing such compounds.

Topics & Concepts

ChemistryCombinatorial chemistryMedicineNeutrophil, Myeloperoxidase and Oxidative MechanismsCell Adhesion Molecules ResearchNF-κB Signaling Pathways