Litcius/Paper detail

Strategies for developing retinoic acid receptor alpha-selective antagonists as novel agents for male contraception

Md Abdullah Al Noman, Rebecca A. D. Cuellar, Jillian L. Kyzer, Sanny S.W. Chung, Narsihmulu Cheryala, Trinh A. D. Holth, Soma Maitra, Tahmina Naqvi, H.L.S. Wong, E. Schönbrunn, Jon E. Hawkinson, Debra J. Wolgemuth, Gunda I. Georg

2023European Journal of Medicinal Chemistry10 citationsDOIOpen Access PDF

Topics & Concepts

ChemistryPharmacologyRetinoic acidSpermatogenesisBioavailabilityTransactivationIn vivoPharmacokineticsOral administrationAntagonistRetinoic acid receptorMale contraceptiveIn vitroReceptorEndocrinologyBiochemistryPopulationBiologyMedicineFamily planningResearch methodologyBiotechnologyEnvironmental healthTranscription factorGeneRetinoids in leukemia and cellular processesEstrogen and related hormone effectsReproductive biology and impacts on aquatic species