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Novel non-covalent LSD1 inhibitors endowed with anticancer effects in leukemia and solid tumor cellular models

Martina Menna, Francesco Fiorentino, Biagina Marrocco, Alessia Lucidi, Stefano Tomassi, Domenica Cilli, Mauro Romanenghi, Matteo Cassandri, Silvia Pomella, Michele Pezzella, Donatella Del Bufalo, Mohammad Salik Zeya Ansari, Nevena Tomašević, Milan Mladenović, Monica Viviano, Gianluca Sbardella, Rossella Rota, Daniela Trisciuoglio, Saverio Minucci, Andrea Mattevi, Dante Rotili, Antonello Mai

2022European Journal of Medicinal Chemistry29 citationsDOIOpen Access PDF

Topics & Concepts

ChemistryCancer cellCell cultureCancer researchDemethylaseCell growthQuinazolineBiochemistryHistoneCancerGeneStereochemistryBiologyGeneticsHistone Deacetylase Inhibitors ResearchEpigenetics and DNA MethylationCancer-related gene regulation
Novel non-covalent LSD1 inhibitors endowed with anticancer effects in leukemia and solid tumor cellular models | Litcius