Litcius/Paper detail

Atorvastatin Potentially Reduces Mycobacterial Severity through Its Action on Lipoarabinomannan and Drug Permeability in Granulomas

Kusuma Sai Davuluri, Amit Kumar Singh, Ajay Vir Singh, Pooja Chaudhary, Sunil Kumar Raman, Shweta Kushwaha, Shoor Vir Singh, Devendra Singh Chauhan

2023Microbiology Spectrum18 citationsDOIOpen Access PDF

Abstract

and an increase in the vascularity at the granuloma site reduce the permeability of rifampicin and isoniazid concentrations. However, very few studies have assessed the effect of statins on drug penetration, which can be increased through a reduction in cholesterol and vascularity. Herein, we used atorvastatin, a 3-hydroxy-3-methylglutaryl coenzyme A (HMG-CoA) reductase inhibitor, to observe its effect on bacterial burden through increasing the drug concentration at the infection site. Our main research goal is to diminish mycobacterial dissemination and attenuate bacterial growth by increasing drug permeability.

Topics & Concepts

AtorvastatinIsoniazidRifampicinTuberculosisMycobacterium tuberculosisPharmacologyMedicineDrugStatinImmunologyMicrobiologyBiologyPathologyInternal medicineTuberculosis Research and EpidemiologyBiochemical and Molecular ResearchComputational Drug Discovery Methods