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Lead discovery, chemical optimization, and biological evaluation studies of novel histone methyltransferase SET7 small-molecule inhibitors

Zeng Hou, Wenjian Min, Rukang Zhang, Ao Niu, Yuan‐Qing Li, Liyuan Cao, Jie Han, Cheng Luo, Peng Yang, Hong Ding

2020Bioorganic & Medicinal Chemistry Letters16 citationsDOIOpen Access PDF

Topics & Concepts

ChemistryMethyltransferaseEpigeneticsHistone H3Histone methyltransferaseHistoneMethylationLead compoundBiochemistryCancer researchIn vitroBiologyGeneEpigenetics and DNA MethylationCancer-related gene regulationRNA modifications and cancer
Lead discovery, chemical optimization, and biological evaluation studies of novel histone methyltransferase SET7 small-molecule inhibitors | Litcius