Novel GPR43 Agonists Exert an Anti-Inflammatory Effect in a Colitis Model
Bi-Oh Park, Jong Soon Kang, Suresh Raj Paudel, Sung Goo Park, Byoung Chul Park, Sang‐Bae Han, Young‐Shin Kwak, Jeong‐Hoon Kim, Sunhong Kim
Abstract
, compound 110 induced more potent attenuation of inflammation. These novel allosteric agonists of GPR43 clearly display anti-inflammatory potential, supporting their clinical utility as therapeutic drugs.
Topics & Concepts
ColitisPharmacologyMedicineTraditional medicineInternal medicineHelicobacter pylori-related gastroenterology studiesGastrointestinal motility and disordersDigestive system and related health