Design, synthesis, and biological evaluation of 1-methyl-1H-pyrazolo[4,3-b]pyridine derivatives as novel small-molecule inhibitors targeting the PD-1/PD-L1 interaction
Xinyan Dai, Ke Wang, Hao Chen, Xupeng Huang, Zhiqiang Feng
Topics & Concepts
ChemistryJurkat cellsSmall moleculeIC50DimerStereochemistryPyridineDocking (animal)Monoclonal antibodyT cellIn vitroBiochemistryAntibodyImmune systemBiologyMedicineImmunologyOrganic chemistryMedicinal chemistryNursingCAR-T cell therapy researchCancer Immunotherapy and BiomarkersMelanoma and MAPK Pathways