Blood-stage antimalarial activity, favourable metabolic stability and in vivo toxicity of novel piperazine linked 7-chloroquinoline-triazole conjugates
Amad Uddin, Sonal Gupta, Rumaisha Shoaib, Babita Aneja, Iram Irfan, Kanika Gupta, Neha Kanwar Rawat, Jill M. Combrinck, Bhumika Kumar, Mohd Aleem, Phool Hasan, Mukesh C. Joshi, Yashpal S. Chhonker, Muhammad Zahid, Afzal Hussain, Kailash C. Pandey, Mohamed F. Alajmi, Daryl J. Murry, Timothy J. Egan, Shailja Singh, Mohammad Abid
Topics & Concepts
ChemistryPharmacologyPlasmodium falciparumChloroquineIn vivoHemozoinTriazoleMalariaToxicityPiperazineBiochemistryHemeBiologyEnzymeImmunologyBiotechnologyOrganic chemistryMalaria Research and ControlHIV/AIDS drug development and treatmentHIV Research and Treatment