Targeted degradation of activating estrogen receptor α ligand-binding domain mutations in human breast cancer
Thomas L. Gonzalez, Molly Hancock, Siqi Sun, Christina L. Gersch, José M. Larios, Wadie David, Jiantao Hu, Daniel F. Hayes, Shaomeng Wang, James M. Rae
Topics & Concepts
Estrogen receptorFulvestrantEstrogen receptor alphaCancer researchBiologyDownregulation and upregulationEstrogenMutantEstrogen receptor betaReceptorMolecular biologyEndocrinologyInternal medicineCancerBreast cancerBiochemistryMedicineGeneticsGeneEstrogen and related hormone effectsProtein Degradation and InhibitorsAdvanced Breast Cancer Therapies