Scaffold Hopping Method for Design and Development of Potential Allosteric AKT Inhibitors
Alireza Poustforoosh
Topics & Concepts
Allosteric regulationScaffoldProtein kinase BChemistryComputational biologyScaffold proteinBiologySignal transductionBiochemistryComputer scienceEnzymeDatabasePI3K/AKT/mTOR signaling in cancerEnzyme function and inhibitionReceptor Mechanisms and Signaling