Discovery of novel fatty acid amide hydrolase (FAAH) inhibitors as anti-Alzheimer’s agents through pharmacophore-based virtual screening, molecular docking and experimental validation
Smita Jain, Swapnil Sharma, Ajita Paliwal, Jaya Dwivedi, Sarvesh Paliwal, Vartika Paliwal, Sarvesh Paliwal, Jaiprakash Sharma, Sarvesh Paliwal, Jaiprakash Sharma
Topics & Concepts
PharmacophoreFatty acid amide hydrolaseChemistryVirtual screeningLipinski's rule of fiveDocking (animal)Drug discoveryPharmacologyAmyloid betaEnzymeBiochemistryStereochemistryIn silicoMedicineCannabinoid receptorGeneReceptorPeptideNursingAgonistCannabis and Cannabinoid ResearchCholinesterase and Neurodegenerative DiseasesPharmacogenetics and Drug Metabolism