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Characterization of SPK 98, a Torin2 analog, as ATR and mTOR dual kinase inhibitor

Rashmi Bhakuni, Althaf Shaik, Bhanu Priya, Sivapriya Kirubakaran

2020Bioorganic & Medicinal Chemistry Letters10 citationsDOI

Topics & Concepts

ChemistryPI3K/AKT/mTOR pathwayKinaseDiscovery and development of mTOR inhibitorsBiochemistryCell culturePharmacologySignal transductionBiologyGeneticsUbiquitin and proteasome pathwaysCell death mechanisms and regulationCancer-related Molecular Pathways
Characterization of SPK 98, a Torin2 analog, as ATR and mTOR dual kinase inhibitor | Litcius