Identification of new [1,2,4]triazolo[4,3-a]quinoxalines as potent VEGFR-2 tyrosine kinase inhibitors: Design, synthesis, anticancer evaluation, and in silico studies
Nawaf A. Alsaif, Mohammed S. Taghour, Mohammed M. Alanazi, Ahmad J. Obaidullah, Wael A. Alanazi, Abdullah F. Alasmari, Hussam Albassam, Mohammed A. Dahab, Hazem A. Mahdy
Topics & Concepts
ChemistryIn silicoTyrosine kinaseStereochemistryKinaseStructure–activity relationshipIn vitroBiochemistryCombinatorial chemistryPharmacologySignal transductionGeneMedicineSynthesis and Biological EvaluationBioactive Compounds and Antitumor AgentsSynthesis and biological activity