High amount of lecithin facilitates oral delivery of a poorly soluble pyrazoloquinolinone ligand formulated in lipid nanoparticles: Physicochemical, structural and pharmacokinetic performances
Jelena R. Mitrović, Branka Divović, Daniel E. Knutson, Miloš Petković, Djordje Djorović, Danijela Randjelović, Vladimir Dobričić, Jelena Đoković, Dominique Jasmin Lunter, James M. Cook, Miroslav M. Savić, Snežana Savić
Topics & Concepts
BioavailabilityDifferential scanning calorimetryChemistryLecithinParticle sizeSolubilityNanoparticlePharmacokineticsChromatographyAqueous solutionOrganic chemistryMaterials scienceNanotechnologyPharmacologyPhysical chemistryMedicineThermodynamicsPhysicsAdvancements in Transdermal Drug DeliveryLipid Membrane Structure and BehaviorDrug Solubulity and Delivery Systems