TLR4 biased small molecule modulators
Cong Lin, Hongshuang Wang, Miyuan Zhang, Sanam Mustafa, Yibo Wang, Hongyuan Li, Hang Yin, Mark R. Hutchinson, Xiaohui Wang
Topics & Concepts
Drug discoveryG protein-coupled receptorReceptorFunctional selectivityTLR4Signal transductionSmall moleculeTRIFBiologyComputational biologyNeurosciencePharmacologyToll-like receptorCell biologyBioinformaticsBiochemistryInnate immune systemReceptor Mechanisms and SignalingImmune Response and InflammationNeuropeptides and Animal Physiology