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Pyrazole and pyrazolone derivatives as specific α-glucosidase inhibitors: in vitro combined with in silico, hemolytic and cytotoxicity studies

Ines Dhouib, Mehdi Messaâd, Basma HadjKacem, Imen Fendri, Hafedh Majdoub, Bassem Khemakhem

2023Journal of Molecular Structure14 citationsDOI

Topics & Concepts

AcarboseChemistryPyrazolePyrazolonePyrazolonesIC50AmylaseIn vitroCytotoxicityStereochemistryPostprandialEnzymeBiochemistryMedicinal chemistryInsulinMedicineEndocrinologyNatural Antidiabetic Agents StudiesEnzyme Production and CharacterizationPsidium guajava Extracts and Applications
Pyrazole and pyrazolone derivatives as specific α-glucosidase inhibitors: in vitro combined with in silico, hemolytic and cytotoxicity studies | Litcius