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Synthetic lethality in cancer drug discovery: challenges and opportunities

Emanuel Gonçalves, Colm J. Ryan, David J. Adams

2025Nature Reviews Drug Discovery11 citationsDOI

Topics & Concepts

Synthetic lethalityDrug discoveryComputational biologyPrioritizationCancer drugsCancerDrug developmentPhenotypic screeningBioinformaticsIdentification (biology)MedicineComputer scienceBiologyMutagenesisCancer treatmentPTENDruggabilityTranslation (biology)DrugPhenotypeLethalityGene deletionPrecision medicineCRISPR and Genetic EngineeringComputational Drug Discovery MethodsCell Image Analysis Techniques
Synthetic lethality in cancer drug discovery: challenges and opportunities | Litcius