Structural analysis of setmelanotide binding to MC4R variants in comparison to wild-type receptor
Maha M. Hammad, Anwar Mohammad, Nada Alam-Eldin, Dhanya Madhu, Fahd Al‐Mulla, Mohamed Abu‐Farha, Jehad Abubaker
Topics & Concepts
Melanocortin 4 receptorAgonistMelanocortin 3 receptorMelanocortinReceptorDocking (animal)Energy homeostasisMissense mutationBiologyWild typeGlucose homeostasisChemistryGeneticsMutationEndocrinologyMelanocortin receptorGeneObesityMutantMedicineInsulin resistanceNursingRegulation of Appetite and ObesityBiochemical Analysis and Sensing TechniquesAdipokines, Inflammation, and Metabolic Diseases