Design, synthesis and biological evaluation of 3-arylisoquinoline derivatives as topoisomerase I and II dual inhibitors for the therapy of liver cancer
Xuemei Deng, Tian Luo, Xi Zhang, Yuehua Li, Liming Xie, Weifan Jiang, Linyi Liu, Zhen Wang
Topics & Concepts
TopoisomeraseChemistryDruggabilityIsoquinolineDNA damageEtoposideCytotoxicityBiochemistryTopotecanStereochemistryDocking (animal)Cancer cellIn vitroDNABiologyCancerGeneticsNursingGeneMedicineChemotherapyCancer therapeutics and mechanismsBerberine and alkaloids researchSynthesis and Biological Activity