Litcius/Paper detail

Synthesis and evaluation of sulfonamide derivatives targeting EGFR790M/L858R mutations and ALK rearrangement as anticancer agents

Longcai Cao, Han Yao, Linlin Yu, Yuanyuan Ren, Jiadai Liu, Xingshu Li, Jia Xian

2023Bioorganic & Medicinal Chemistry12 citationsDOIOpen Access PDF

Topics & Concepts

ChemistryCell cultureCytotoxicitySulfonamideApoptosisCell growthMolecular biologyBiochemistryCancer researchStereochemistryIn vitroBiologyGeneticsLung Cancer Treatments and MutationsCancer therapeutics and mechanismsPI3K/AKT/mTOR signaling in cancer