Significance of Basal Membrane Permeability of Epithelial Cells in Predicting Intestinal Drug Absorption
Aoi Yoshitomo, Satoshi Asano, Shizuka Hozuki, Yuta Tamemoto, Yukihiro Shibata, Natsumi Hashimoto, Keita Takahashi, Yoko Sasaki, Naoka Ozawa, Michiharu Kageyama, Takeshi Iijima, Yasuhiro Kazuki, Hiromi Sato, Akihiro Hisaka
Topics & Concepts
Paracellular transportP-glycoproteinChemistryPharmacokineticsEffluxMediated transportTranscellularIntracellularPassive transportPermeability (electromagnetism)Apical membraneCaco-2QuinidineMembrane transportMetabolismPharmacologyMembraneBiochemistryBiologyCellMultiple drug resistanceAntibioticsDrug Transport and Resistance MechanismsPharmacological Effects and Toxicity StudiesPharmacogenetics and Drug Metabolism