Synthesis and biological evaluation of acridine-based histone deacetylase inhibitors as multitarget agents against Alzheimer’s disease
Hui-Ju Tseng, Mei-Hsiang Lin, Young‐Ji Shiao, Ying-Chen Yang, Jung-Chun Chu, Chun-Yung Chen, Yi‐Ying Chen, Tony Eight Lin, Chih-Jou Su, Shiow‐Lin Pan, Liang‐Chieh Chen, Chen‐Yu Wang, Kai‐Cheng Hsu, Wei‐Jan Huang
Topics & Concepts
ChemistryHistone deacetylaseAcridineAcridine derivativesPharmacologyBiological activityHistone deacetylase inhibitorAlzheimer's diseaseBiochemistryHistoneDiseaseStereochemistryIn vitroOrganic chemistryInternal medicineGeneMedicineHistone Deacetylase Inhibitors ResearchCholinesterase and Neurodegenerative DiseasesSynthesis and Characterization of Pyrroles