Discovery of 4-(3,5-dimethoxy-4-(((4-methoxyphenethyl)amino)methyl)phenoxy)-N-phenylaniline as a novel c-myc inhibitor against colorectal cancer in vitro and in vivo
Jie Yang, Chao-Guo Cao, Dan Luo, Suke Lan, Meng Luo, Huifang Shan, Xinyu Ma, Yuanyuan Liu, Su Yu, Xin-Xin Zhong, Rui Li
Topics & Concepts
ChemistryCytotoxicityIn vivoColorectal cancerApoptosisIC50OncogeneMTT assayDownregulation and upregulationCancerIn vitroToxicityCancer researchWestern blotPharmacologyMolecular biologyBiochemistryCell cycleBiologyMedicineInternal medicineOrganic chemistryGeneBiotechnologyCancer therapeutics and mechanismsSynthesis and biological activityQuinazolinone synthesis and applications