Targeted selective degradation of Bruton’s tyrosine kinase by PROTACs
Shaodong Liu, Yang Da, Feng Wang, Renjie Yan, Yongzhi Shu, Pei Lin, Jun Lin
Topics & Concepts
Bruton's tyrosine kinaseChemistryIbrutinibTyrosine kinasePharmacologyCancer researchIn vivoProtein degradationKinaseProteasomeBiochemistrySignal transductionImmunologyBiologyLeukemiaBiotechnologyChronic lymphocytic leukemiaProtein Degradation and InhibitorsMultiple Myeloma Research and TreatmentsChronic Lymphocytic Leukemia Research