A small-molecule activation mechanism that directly opens the KCNQ2 channel
Shao-ying Zhang, Demin Ma, Kun Wang, Ya Li, Zhenni Yang, Xiaoxiao Li, Junnan Li, Jiangnan He, Lianghe Mei, Yangliang Ye, Zongsheng Chen, Juwen Shen, Panpan Hou, Jiangtao Guo, Qiansen Zhang, Huaiyu Yang
Topics & Concepts
GatingPotassium channelIon channelChemistryActivator (genetics)Voltage-gated ion channelConductanceMechanism (biology)BiophysicsDrug discoverySmall moleculeVoltage-gated potassium channelNanotechnologyMaterials scienceBiochemistryBiologyPhysicsGeneReceptorCondensed matter physicsQuantum mechanicsIon channel regulation and functionCardiac electrophysiology and arrhythmiasElectrochemical Analysis and Applications