Hetero-aryl bromide precursor fluorine-18 radiosynthesis and preclinical evaluation of a novel positron emission tomography (PET) tracer [18F]GSK1482160
Guolong Huang, Xiaolei Lu, Yifan Qiu, Lei Bi, Peizhen Ye, Min Yang, Yanfang Shen, Hongjun Jin, Junbin Han
Topics & Concepts
RadiosynthesisChemistryBiodistributionRadioligandPositron emission tomographyIn vivoBromideEx vivoPurinergic receptorRadiochemistryPet imagingTranslocator proteinBlood–brain barrierNuclear medicineIn vitroExtracellularBiochemistryMicrogliaCentral nervous systemInternal medicineInflammationOrganic chemistryBiologyMedicineBiotechnologyAdenosine and Purinergic SignalingSynthesis and Biological EvaluationPharmacological Receptor Mechanisms and Effects