<i>In vitro</i> anti-TB properties, <i>in silico</i> target validation, molecular docking and dynamics studies of substituted 1,2,4-oxadiazole analogues against <i>Mycobacterium tuberculosis</i>
Pran Kishore Deb, Nizar A. Al‐Shar’i, Katharigatta N. Venugopala, Melendhran Pillay, Pobitra Borah
Abstract
, promising leads worthy of further optimisation.
Topics & Concepts
In silicoMycobacterium tuberculosisDocking (animal)OxadiazoleIn vitroChemistryComputational biologyMolecular dynamicsStereochemistryTuberculosisCombinatorial chemistryBiologyBiochemistryComputational chemistryMedicineOrganic chemistryPathologyGeneNursingSynthesis and biological activityComputational Drug Discovery MethodsTuberculosis Research and Epidemiology