Targeting glutaminase 1 (GLS1) by small molecules for anticancer therapeutics
Yangyang Chen, Lun Tan, Jing Gao, Congcong Lin, Fengbo Wu, Yang Li, Jifa Zhang
Topics & Concepts
Allosteric regulationSmall moleculeGlutaminaseChemistryDruggabilityCancerIn vivoDrug discoveryCancer cellComputational biologyCancer researchEnzymeBiochemistryBiologyGlutamineGeneAmino acidBiotechnologyGeneticsCancer, Hypoxia, and MetabolismEpigenetics and DNA MethylationRNA modifications and cancer