Design, synthesis, and biological evaluation of low-toxic lappaconitine derivatives as potential analgesics
Yuzhu Li, Yu-Shan Shang, Xiaohuan Li, Yinyong Zhang, Jiang Xie, Lin Chen, Feng Gao, Xian‐Li Zhou
Topics & Concepts
ChemistryAnalgesicToxicityPharmacologyMetaboliteLead compoundAcute toxicityIn vivohERGAlkaloidStereochemistryBiochemistryIn vitroPotassium channelOrganic chemistryMedicineBiotechnologyEndocrinologyBiologyPlant-based Medicinal ResearchBerberine and alkaloids researchBioactive Natural Diterpenoids Research