Discovery of a miniaturized PROTAC with potent activity and high selectivity
Lidong Gong, Ridong Li, Jingjing Gong, Xianling Ning, Jiawei Sun, Qiang Ma, Chuanda Zhu, Yuanyuan Yang, Kerui Lin, Yanglonghao Li, Qiang Zhang, Tiancheng Li, Zhiqiang Lin, Qiang Zhang, Tiancheng Li, Zhiqiang Lin
Topics & Concepts
Anaplastic lymphoma kinaseCeritinibChemistryMutantSmall moleculeDrug discoveryALK inhibitorAlectinibDrugCombinatorial chemistryCancer researchComputational biologyPharmacologyBiochemistryGeneBiologyMedicineLung cancerOncologyMalignant pleural effusionProtein Degradation and InhibitorsPeptidase Inhibition and AnalysisMultiple Myeloma Research and Treatments