Litcius/Paper detail

Development of STING degrader with double covalent ligands

Miki Nakamura, Nobumichi Ohoka, Norihito Shibata, Takao Inoué, Genichiro Tsuji, Yosuke Demizu

2024Bioorganic & Medicinal Chemistry Letters10 citationsDOI

Topics & Concepts

StingStimulator of interferon genesChemistryEndoplasmic reticulumUbiquitin ligaseCovalent bondUbiquitinInnate immune systemLigand (biochemistry)ProteolysisReceptorCell biologyPharmacologyBiochemistryMedicineBiologyGeneEnzymeEngineeringOrganic chemistryAerospace engineeringinterferon and immune responsesUbiquitin and proteasome pathwaysNF-κB Signaling Pathways
Development of STING degrader with double covalent ligands | Litcius