Design and synthesis of potent PAR-1 antagonists based on vorapaxar
Mengna Fan, Min Han, Yan Xia, Yingbin Zhang, Yang Chu, Guirong Bai, Wei Li, Ju Li, Lihui Zhao, Yi He, Xiaohui Ma, Zhongyu Duan
Topics & Concepts
ChemistryAntagonistIC50PharmacologyInhibitory postsynaptic potentialPharmacokineticsPotencyIntracellularStereochemistryIn vitroReceptorBiochemistryEndocrinologyMedicineBlood Coagulation and Thrombosis MechanismsAntiplatelet Therapy and Cardiovascular DiseasesAcute Myocardial Infarction Research