Pregnancy-Related Hormones Increase Nifedipine Metabolism in Human Hepatocytes by Inducing CYP3A4 Expression
Raju Khatri, Natasha Kulick, Rebecca J.B. Rementer, John K. Fallon, Craig Sykes, Amanda P. Schauer, Melina M. Malinen, Merrie Mosedale, Paul B. Watkins, Angela D. M. Kashuba, Kim Boggess, Philip C. Smith, Kim L. R. Brouwer, Craig R. Lee
Topics & Concepts
CYP3A4NifedipineHepatocyteMetabolismCytochrome P450EndocrinologyInternal medicineDrug metabolismIsozymeChemistryMifepristoneBiologyEnzymeBiochemistryPregnancyIn vitroMedicineCalciumGeneticsPregnancy and preeclampsia studiesPregnancy and Medication ImpactPharmacological Effects and Toxicity Studies