Inhibitory activity on cholinesterases produced by aryl-phthalimide derivatives: green synthesis, in silico and in vitro evaluation
Omar Ruiz-Maciel, Itzia I. Padilla‐Martínez, Luis A. Sánchez‐Labastida, Marvin A. Soriano‐Ursúa, Erik Andrade‐Jorge, José G. Trujillo‐Ferrara
Topics & Concepts
ButyrylcholinesteraseAcetylcholinesteraseChemistryAchéIn silicoPhthalimideCholinesteraseIn vitroIC50PharmacologyEnzymeBiochemistryMedicineGeneCholinesterase and Neurodegenerative DiseasesComputational Drug Discovery MethodsChemical synthesis and alkaloids