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Structure-based identification of new orally bioavailable BRD9-PROTACs for treating acute myelocytic leukemia

Jingyu Zhang, Haiting Duan, Renzhao Gui, Mingfei Wu, Liteng Shen, Yuheng Jin, Ao Pang, Xiaoli Yu, Shenxin Zeng, Bo Zhang, Nengming Lin, Wenhai Huang, Yuwei Wang, Xiaojun Yao, Jia Li, Xiaowu Dong, Yubo Zhou, Jinxin Che

2023European Journal of Medicinal Chemistry14 citationsDOI

Topics & Concepts

ChemistryPharmacologyBioavailabilityMedicineProtein Degradation and InhibitorsMultiple Myeloma Research and TreatmentsPeptidase Inhibition and Analysis
Structure-based identification of new orally bioavailable BRD9-PROTACs for treating acute myelocytic leukemia | Litcius