In silico studies of 2-aryloxy-1,4- naphthoquinone derivatives as antibacterial agents against Escherichia coli using 3D-QSAR, ADMET properties, molecular docking, and molecular dynamics
Khaoula Mkhayar, Rachid Haloui, Ossama Daouı, Kaouakeb Elkhattabi, Samir Chtita, Souad Elkhattabi
Topics & Concepts
Quantitative structure–activity relationshipIn silicoMolecular dynamicsChemistryDocking (animal)Molecular modelComputational chemistryNaphthoquinoneEscherichia coliCombinatorial chemistryComputational biologyStereochemistryBiologyBiochemistryOrganic chemistryGeneMedicineNursingBioactive Compounds and Antitumor AgentsComputational Drug Discovery MethodsSynthesis and biological activity